Tiapride

  • N-[2-(Ethylamino)ethyl]-2-methoxy-5-(methylsulfonyl)benzamide
  • N-[2-(Diethylamino)ethyl]-2-methoxy-5-(methylsulfonyl)benzamide
Formula
C15H24N2O4S . HCl
Structure
Uses
D2 and D3 dopamine receptor antagonist; antipsychotic.

Registry Numbers and Inventories.
CAS
51012-32-9
EC (EINECS/ELINCS)
256-907-9
RTECS
CV4203700
RTECS class
Reproductive Effector
Merck
12,9561
Beilstein/Gmelin
2390588
Beilstein Reference
6-10

Properties.
Formula
C15H24N2O4S . HCl
Formula mass
328.43
Melting point, °C
120
Boiling point, °C
498
Vapor pressure, mmHg
5E-10 (25 C)
Solubility in water
Soluble
pKa/pKb
4.40 (pKb)
Heat of vaporization
76.6 kJ/mol

Hazards and Protection.
Storage
Store at 2-8 C.
Protection
Wear appropriate government approved respirator, chemical-resistant gloves, safety goggles, other protective clothing.
Small spills/leaks
Sweep up, place in a bag and hold for waste disposal. Avoid raising dust. Ventilate area and wash spill site after material pickup is complete.
Stability
Stable at normal temperatures and pressures.
Decomposition
Carbon monoxide, Carbon dioxide, Nitrogen oxides, Sulfur oxides.

Fire.
Flash Point,°C
255
Fire fighting
Extinguish using Water spray. Carbon dioxide, dry chemical powder, or appropriate foam. Wear self-contained breathing apparatus and protective clothing to prevent contact with skin and eyes.
Hazards
Emits toxic fumes under fire conditions.

Health.
Exposure effects
Avoid contact and inhalation.

First aid
 
   Ingestion
If swallowed, wash out mouth with water provided person is conscious. Call a physician.
   Inhalation
If inhaled, remove to fresh air. If breathing becomes difficult, call a physician.
   Skin
In case of skin contact, flush with copious amounts of water for at least 15 minutes. Remove contaminated clothing and shoes. Call a physician.
   Eyes
In case of contact with eyes, flush with copious amounts of water for at least 15 minutes. Assure adequate flushing by separating the eyelids with fingers. Call a physician.

Transport.